The Organic chemistry of drug design and drug action - Silverman, Richard B. (New Delhi Elsevier Academic Press, 2012)
Introduction -- Drug discovery, design, and development -- Receptors -- Enzymes -- Enzyme inhibition and inactivation -- DNA-interactive agents -- Drug metabolism -- Prodrugs and drug delivery systems.
Keywords: Drugs - Design -- Drugs - Metabolism -- Chemistry, Pharmaceutical -- Chemistry, Organic